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Table 2 IC50 values for inhibition of cell proliferation

From: High basal Wnt signaling is further induced by PI3K/mTor inhibition but sensitive to cSRC inhibition in mammary carcinoma cell lines with HER2/3 overexpression

Inhibitor

IC50 proliferation

Concentration used

References

 

CIPm

CMT -U27

  

BEZ235

69 nM

29 nM

50 nM

[33, 34]

Everolimus

3 nM

1 nM

100 nM

[35]

Src-I1

4 μM

1 μM

20 μM

[49]