From: Role of drug transporters and drug accumulation in the temporal acquisition of drug resistance
Dose | Doxorubicin | Epirubicin | Paclitaxel | Docetaxel |
---|---|---|---|---|
IC50 | 8.91 nM | 4.79 nM | 0.56 nM | 0.51 nM |
1 | 8.91 pM | 4.79 pM | 0.56 pM | 0.51 pM |
2 | 26.7 pM | 14.4 pM | 1.67 pM | 1.52 pM |
3 | 80.1 pM | 43.2 pM | 5.01 pM | 4.56 pM |
4 | 240 pM | 130 pM | 15.0 pM | 13.7 pM |
5 | 720 pM | 390 pM | 45.0 pM | 41.1 pM |
6 | 2.16 nM | 1.17 nM | 135 pM | 123 pM |
7 | 6.48 nM | 3.51 nM | 405 pM | 369 pM |
8 | 19.4 nM | 10.5 nM | 1.22 nM | 1.11 nM |
9 | 29.1 nM | 31.5 nM | 3.66 nM | 3.33 nM |
10 | 43.6 nM | 94.5 nM | 11.0 nM | 5.00 nM |
11 | 65.4 nM | 284 nM | 33.0 nM | 15.0 nM |
12 | 98.1 nM* | 852 nM | 99.0 nM | 45.0 nM* |