From: Protein kinase C-delta inactivation inhibits the proliferation and survival of cancer stem cells in culture and in vivo
Generation
PKCδIC50
PKCαIC50
PKCδ/PKCα
Selectivity ratio
1
3 μM
75 μM
28-fold
2
2 μM
157 μM
56-fold
3
0.05 μM
50 μM
1000-fold