From: Antagonists of the serotonin receptor 5A target human breast tumor initiating cells
Compound | Cell Line | IC50 (μM) | |
---|---|---|---|
Sphere Formation | PrestoBlue Reduction | ||
SB-699551 | HCC1954 | 0.3 | 0.2 |
MCF-7 | 0.2 | 0.2 | |
G1A-(S) | HCC1954 | 2.5 | 6.7 |
MCF-7 | 2.5 | 3.0 | |
G1A-(R) | HCC1954 | 16.4 | 14.2 |
MCF-7 | 11.0 | 21.9 | |
G1B-(S) | HCC1954 | 3.0 | 3.8 |
MCF-7 | 2.2 | 1.3 | |
G1B-(R) | HCC1954 | 11.3 | 11.8 |
MCF-7 | 11.4 | 14.1 | |
AS2030680 | HCC1954 | 1.8 | 3.9 |
MCF-7 | 2.0 | 5.6 | |
ASP5736 | HCC1954 | > 25.0 | > 25.0 |
MCF-7 | > 25.0 | > 25.0 |