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Table 1 Calcitonin family of receptors [10, 11, 38]

From: Expression and activity of the calcitonin receptor family in a sample of primary human high-grade gliomas

Receptor

Heteromers

Peptides rank order of potency (human)

CTR

CTR

sCT ≥ hCT > AMY, αCGRP > AM, intermedin

AMY1

CTR + RAMP1

sCT ≥ AMY ≥ αCGRP > intermedin ≥ hCT > AM

AMY2

CTR + RAMP2

Poorly defined

AMY3

CTR + RAMP3

sCT ≥ AMY > αCGRP > intermedin ≥ hCT > AM

CGRP

CLR + RAMP1

αCGRP > AM ≥ intermedin > AMY ≥ sCT

AM1

CLR + RAMP2

AM > intermedin > α-CGRP, AMY > sCT

AM2

CLR + RAMP3

AM ≥ intermedin ≥ α-CGRP > AMY > SCT

  1. Rank order of potency for endogenous peptide ligands for calcitonin receptor family of receptors. sCT Salmon CT, hCT Human CT, AMY1 Amylin 1 receptor, AMY2 Amylin 2 receptor, AMY3 Amylin 3 receptor, CGRP Calcitonin gene related peptide receptor