Receptor | Heteromers | Peptides rank order of potency (human) |
---|---|---|
CTR | CTR | sCT ≥ hCT > AMY, αCGRP > AM, intermedin |
AMY1 | CTR + RAMP1 | sCT ≥ AMY ≥ αCGRP > intermedin ≥ hCT > AM |
AMY2 | CTR + RAMP2 | Poorly defined |
AMY3 | CTR + RAMP3 | sCT ≥ AMY > αCGRP > intermedin ≥ hCT > AM |
CGRP | CLR + RAMP1 | αCGRP > AM ≥ intermedin > AMY ≥ sCT |
AM1 | CLR + RAMP2 | AM > intermedin > α-CGRP, AMY > sCT |
AM2 | CLR + RAMP3 | AM ≥ intermedin ≥ α-CGRP > AMY > SCT |