Name | Solvent | |
---|---|---|
Dasatinib | DMSO | ABL, PDGFR, KIT, SRC |
Erlotinib | DMSO | EGFR |
Gefitinib | DMSO | EGFR |
Imatinib | DMSO | ABL, PDGFR, KIT |
Masitinib | DMSO | c-KIT, PDGFRα, −β, Lyn, FGFR3, FAK pathway |
Nilotinib | DMSO | ABL, PDGFR, KIT |
Toceranib | DMSO | VEGFR2, PDGFRβ, c-KIT |
Sorafenib | DMSO | VEGFR2, PDGFR, KIT, FLT3, BRAF |
Sunitinib | DMSO | VEGFR, KIT, PDGFR, RET, CSF1R, FLT3 |
Tozasertib | DMSO | SRC, GSK3, FLT3, JAK2, BCR-ABL |
CCNU | Ethanol | Alkylation and cross-linking of DNA |
Cladribine | DMSO | Purine analogue |
Doxorubicin | Saline | Inhibits DNA topoisomerase II, induces DNA damage and apoptosis |