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Table 2 Kinase panel assay

From: Novel c-Met inhibitor suppresses the growth of c-Met-addicted gastric cancer cells

 

KRC-00715 @ 1 μM

 

KRC-00715 @ 1 μM

 

KRC-00715 @ 1 μM

Abl

104

Fer

100

Lyn

99

Ack1

96

Fes

97

Mer

105

ALK

101

FGFR1

107

Met

−2

Axl

107

Fgr

113

MuSK

106

Blk

102

Flt1

115

PDGFRα

121

Brk

96

Flt3

94

Ret

110

BTK

108

Fms

108

Ron

107

c-Ket

101

Fyn

106

Ros

115

CSK

116

Hck

81

Syk

110

DDR1

90

IGF-1R

92

Tie2

116

EGFR

111

IR

119

TrkA

99

EphA1

117

IRR

90

Yes

114

EphB1

104

JAK1

111

  

FAK

105

KDR

110

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