Substrate/Inhibitor | ||||
---|---|---|---|---|
cell line | L-Glu (μM) IC50[pIC50 ± S.E.M.] | UCPH (μM) IC50[pIC50 ± S.E.M.] | TBOA (μM) IC50[pIC50 ± S.E.M.] | Basal Uptake [% of parental] |
HCT116-PAR | 21 [4.67 ± 0.04] | >100 [<4.0] | 1.8 [5.75 ± 0.03] | 100 |
HCT116-SN38 | 21 [4.67 ± 0.01] | >100 [<4.0] | 1.5 [5.83 ± 0.08] | 40 ± 1.8*** |
HCT116-Oxa | 21 [4.67 ± 0.01] | >100 [<4.0] | 1.5 [5.75 ± 0.08] | 73 ± 6.9* |
LoVo-PAR | 26 [4.59 ± 0.04] | >100 [<4.0] | 1.4 [5.84 ± 0.03] | 100 |
LoVo-SN38 | 28 [4.54 ± 0.10] | >100 [<4.0] | 1.9 [5.83 ± 0.11] | 275 ± 35** |
LoVo-Oxa | 23 [4.64 ± 0.06] | >100 [<4.0] | 2.7 [5.75 ± 0.03] | 97 ± 8.0 NS |